Stereo- and regioselective glycosylation of 4-deoxy-epsilon-rhodomycinone

Filip S. Ekholm; Lucas Lagerquist; Reko Leino

doi:10.1016/j.carres.2011.01.028

Stereo- and regioselective glycosylation of 4-deoxy-epsilon-rhodomycinone

Filip S. Ekholm
, Lucas Lagerquist
, Reko Leino

Forskningsoutput: Tidskriftsbidrag › Artikel › Vetenskaplig › Peer review

2 Citeringar (Scopus)

Sammanfattning

A method for the glycosylation of anthracyclines featuring benzoylated imidate donors has been developed and utilized in the synthesis of glycosylated 4-deoxy-epsilon-rhodomycinone derivatives. Due to its high efficiency, regioselectivity, stereoselectivity, and operational simplicity, the method should prove valuable to researchers working with glycosylation of tetracyclic compounds. (C) 2011 Elsevier Ltd. All rights reserved.

Originalspråk	Odefinierat/okänt
Sidor (från-till)	858–862
Antal sidor	5
Tidskrift	Carbohydrate Research
Volym	346
Nummer	6
DOI	https://doi.org/10.1016/j.carres.2011.01.028
Status	Publicerad - 2011
MoE-publikationstyp	A1 Tidskriftsartikel-refererad

Nyckelord

Anthracycline
Glycosylation
Regioselectivite synthesis
Rhodomycinone glycosides
Stereoselective synthesis

Åtkomst av dokument

10.1016/j.carres.2011.01.028

Citera det här

@article{a6c8931223b84f0d87a080d6454d3d6a,

title = "Stereo- and regioselective glycosylation of 4-deoxy-epsilon-rhodomycinone",

abstract = "A method for the glycosylation of anthracyclines featuring benzoylated imidate donors has been developed and utilized in the synthesis of glycosylated 4-deoxy-epsilon-rhodomycinone derivatives. Due to its high efficiency, regioselectivity, stereoselectivity, and operational simplicity, the method should prove valuable to researchers working with glycosylation of tetracyclic compounds. (C) 2011 Elsevier Ltd. All rights reserved.",

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author = "Ekholm, \{Filip S.\} and Lucas Lagerquist and Reko Leino",

year = "2011",

doi = "10.1016/j.carres.2011.01.028",

language = "Odefinierat/ok{\"a}nt",

volume = "346",

pages = "858–862",

journal = "Carbohydrate Research",

issn = "0008-6215",

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TY - JOUR

T1 - Stereo- and regioselective glycosylation of 4-deoxy-epsilon-rhodomycinone

AU - Ekholm, Filip S.

AU - Lagerquist, Lucas

AU - Leino, Reko

PY - 2011

Y1 - 2011

N2 - A method for the glycosylation of anthracyclines featuring benzoylated imidate donors has been developed and utilized in the synthesis of glycosylated 4-deoxy-epsilon-rhodomycinone derivatives. Due to its high efficiency, regioselectivity, stereoselectivity, and operational simplicity, the method should prove valuable to researchers working with glycosylation of tetracyclic compounds. (C) 2011 Elsevier Ltd. All rights reserved.

AB - A method for the glycosylation of anthracyclines featuring benzoylated imidate donors has been developed and utilized in the synthesis of glycosylated 4-deoxy-epsilon-rhodomycinone derivatives. Due to its high efficiency, regioselectivity, stereoselectivity, and operational simplicity, the method should prove valuable to researchers working with glycosylation of tetracyclic compounds. (C) 2011 Elsevier Ltd. All rights reserved.

KW - Anthracycline

KW - Glycosylation

KW - Regioselectivite synthesis

KW - Rhodomycinone glycosides

KW - Stereoselective synthesis

KW - Anthracycline

KW - Glycosylation

KW - Regioselectivite synthesis

KW - Rhodomycinone glycosides

KW - Stereoselective synthesis

KW - Anthracycline

KW - Glycosylation

KW - Regioselectivite synthesis

KW - Rhodomycinone glycosides

KW - Stereoselective synthesis

U2 - 10.1016/j.carres.2011.01.028

DO - 10.1016/j.carres.2011.01.028

M3 - Artikel

SN - 0008-6215

VL - 346

SP - 858

EP - 862

JO - Carbohydrate Research

JF - Carbohydrate Research

IS - 6

ER -