A Monocarbonyl Curcuminoid Derivative Inhibits the Activity of Human Glutathione Transferase A4-4 and Chemosensitizes Glioblastoma Cells to Temozolomide

Steliana Tsouri, Evanthia Tselo, Georgios E. Premetis, Veronika Furlan, Panagiota D. Pantiora, Barbara Mavroidi, Dimitris Matiadis, Maria Pelecanou, Anastassios C. Papageorgiou, Urban Bren, Marina Sagnou, Nikolaos E. Labrou

Research output: Contribution to journalArticleScientificpeer-review

3 Citations (Scopus)
Original languageEnglish
Article number365
Number of pages18
JournalPharmaceuticals
Volume17
Issue number3
DOIs
Publication statusPublished - Mar 2024
MoE publication typeA1 Journal article-refereed

Keywords

  • GST inhibition
  • Chemoresistance
  • Chemosensitization
  • Curcumin
  • Ellagic acid
  • Glioblastoma
  • human glutathione transferase A4-4
  • Monocarbonyl curcumin derivatives
  • Temozolomide sensitization

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